BIOMAT Database Logo BIOMAT Database Logo

Enkephalin analogs with enhanced opiate activity. 1976

S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf

UI MeSH Term Description Entries
D009294 Narcotics Agents that induce NARCOSIS. Narcotics include agents that cause somnolence or induced sleep (STUPOR); natural or synthetic derivatives of OPIUM or MORPHINE or any substance that has such effects. They are potent inducers of ANALGESIA and OPIOID-RELATED DISORDERS. Analgesics, Narcotic,Narcotic Analgesics,Narcotic,Narcotic Effect,Narcotic Effects,Effect, Narcotic,Effects, Narcotic
D009842 Oligopeptides Peptides composed of between two and twelve amino acids. Oligopeptide
D001923 Brain Chemistry Changes in the amounts of various chemicals (neurotransmitters, receptors, enzymes, and other metabolites) specific to the area of the central nervous system contained within the head. These are monitored over time, during sensory stimulation, or under different disease states. Chemistry, Brain,Brain Chemistries,Chemistries, Brain
D000818 Animals Unicellular or multicellular, heterotrophic organisms, that have sensation and the power of voluntary movement. Under the older five kingdom paradigm, Animalia was one of the kingdoms. Under the modern three domain model, Animalia represents one of the many groups in the domain EUKARYOTA. Animal,Metazoa,Animalia
D001681 Biological Assay A method of measuring the effects of a biologically active substance using an intermediate in vivo or in vitro tissue or cell model under controlled conditions. It includes virulence studies in animal fetuses in utero, mouse convulsion bioassay of insulin, quantitation of tumor-initiator systems in mouse skin, calculation of potentiating effects of a hormonal factor in an isolated strip of contracting stomach muscle, etc. Bioassay,Assay, Biological,Assays, Biological,Biologic Assay,Biologic Assays,Assay, Biologic,Assays, Biologic,Bioassays,Biological Assays
D013329 Structure-Activity Relationship The relationship between the chemical structure of a compound and its biological or pharmacological activity. Compounds are often classed together because they have structural characteristics in common including shape, size, stereochemical arrangement, and distribution of functional groups. Relationship, Structure-Activity,Relationships, Structure-Activity,Structure Activity Relationship,Structure-Activity Relationships
D051381 Rats The common name for the genus Rattus. Rattus,Rats, Laboratory,Rats, Norway,Rattus norvegicus,Laboratory Rat,Laboratory Rats,Norway Rat,Norway Rats,Rat,Rat, Laboratory,Rat, Norway,norvegicus, Rattus

Related Publications

S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf
Structure-activity relationships of enkephalin analogs at opiate and enkephalin receptors: correlation with analgesia.
April 1980, European journal of pharmacology,
S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf
Interaction of S-activated enkephalin analogs with opiate receptors.
December 1989, Biochemistry international,
S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf
Synthesis of two enzyme resistant enkephalin analogs possessing enhanced analgesic activity.
April 1978, Research communications in chemical pathology and pharmacology,
S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf
A cyclic enkephalin analog with high in vitro opiate activity.
December 1980, Proceedings of the National Academy of Sciences of the United States of America,
S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf
Opiate-like peptides. Part XI. 2-[2-phenyl-1,3-indandionyl]--amides of enkephalin analogs. Synthesis and analgesic activity.
January 1988, Polish journal of pharmacology and pharmacy,
S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf
Inactivation of the opiate receptor in bovine caudate nucleus by azide enkephalin analogs.
August 1980, The Journal of biological chemistry,
S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf
Opiate-like peptides. Part XIII. Synthesis and analgesic activity of met-enkephalin analogs substituted in position 4 with D-4-halogenophenylalanine.
January 1991, Polish journal of pharmacology and pharmacy,
S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf
Correlation between pharmacological and opiate receptor binding activities of tetrapeptide acylhydrazide analogs of enkephalin.
July 1981, European journal of pharmacology,
S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf
Dehydro-enkephalins. IV. Discriminative recognition of delta and mu opiate receptors by enkephalin analogs.
January 1982, Biochemical and biophysical research communications,
S Bajusz, and A Z Rónai, and J I Székely, and Z Dunai-Kovács, and I Berzétei, and L Gráf
Acetaldehyde-enkephalins: pronounced changes in the opiate activity of methionine-enkephalin and leucine-enkephalin on reaction with acetaldehyde.
April 1980, FEBS letters,
Copied contents to your clipboard!