Capillary gas chromatographic behaviour of tert.-hydroxylated steroids by trialkylsilylation. 2001

T Iida, and M Hikosaka, and J Goto, and T Nambara
Department of Chemistry, College of Humanities and Sciences, Nihon University, Sakurajousui, Tokyo, Japan. takaiida@chs.nihon-u.ac.jp

Capillary gas chromatographic behaviour was studied for a variety of structurally different bile acids and sterols having one to two tert.-hydroxy groups, together with several sec.-hydroxy groups, at positions C-3, -5, -7, -12, -14, -17, -20, -24, and/or -25. The tert.-hydroxylated steroids were subjected to trimethylsilylation with hexamethyldisilazane/trimethylchlorosilane /pyridine and N,O-bis(trimethylsilyl)acetamide/N-trimethylsilylimidazole/trimethylchlorosilane, and dimethylethylsilylation with N,N,-dimethylethylsilylimidazole. The methylene unit values of the resulting trialkylsilylation products were used for determining their structures of partially and/or fully derivatised ethers. The reactivity of the trialkylsilylation of tert.-hydroxy groups was found to be significantly dependent not only on the derivatisation reagents and conditions used, but also on the position and steric factor of the tert.-hydroxy groups. The following general order of the decreasing reactivity of tert.-hydroxy groups in steroids by trialkylsilyl etherification was observed: 25>20, 24>5beta>17alpha>>14alpha.

UI MeSH Term Description Entries
D002849 Chromatography, Gas Fractionation of a vaporized sample as a consequence of partition between a mobile gaseous phase and a stationary phase held in a column. Two types are gas-solid chromatography, where the fixed phase is a solid, and gas-liquid, in which the stationary phase is a nonvolatile liquid supported on an inert solid matrix. Chromatography, Gas-Liquid,Gas Chromatography,Chromatographies, Gas,Chromatographies, Gas-Liquid,Chromatography, Gas Liquid,Gas Chromatographies,Gas-Liquid Chromatographies,Gas-Liquid Chromatography
D006900 Hydroxylation Placing of a hydroxyl group on a compound in a position where one did not exist before. (Stedman, 26th ed) Hydroxylations
D012794 Sialic Acids A group of naturally occurring N-and O-acyl derivatives of the deoxyamino sugar neuraminic acid. They are ubiquitously distributed in many tissues. N-Acetylneuraminic Acids,Acids, N-Acetylneuraminic,Acids, Sialic,N Acetylneuraminic Acids
D013256 Steroids A group of polycyclic compounds closely related biochemically to TERPENES. They include cholesterol, numerous hormones, precursors of certain vitamins, bile acids, alcohols (STEROLS), and certain natural drugs and poisons. Steroids have a common nucleus, a fused, reduced 17-carbon atom ring system, cyclopentanoperhydrophenanthrene. Most steroids also have two methyl groups and an aliphatic side-chain attached to the nucleus. (From Hawley's Condensed Chemical Dictionary, 11th ed) Steroid,Catatoxic Steroids,Steroids, Catatoxic
D015394 Molecular Structure The location of the atoms, groups or ions relative to one another in a molecule, as well as the number, type and location of covalent bonds. Structure, Molecular,Molecular Structures,Structures, Molecular

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