Stability of an extemporaneously compounded clonidine hydrochloride oral liquid. 1992

M L Levinson, and C E Johnson
Pharmacy Department, University Medical Center, Tucson, AZ.

The stability of clonidine hydrochloride in an extemporaneous oral liquid formulation refrigerated for 28 days was studied. A suspension was prepared by grinding commercially available 0.2-mg clonidine hydrochloride tablets, adding Purified Water, USP, to form a paste, and then adding Simple Syrup, NF. A control solution was prepared from analytical grade clonidine hydrochloride powder in Simple Syrup, NF. The final concentration of clonidine hydrochloride in both formulations was 0.1 mg/mL. Three samples of each preparation were stored in 2-ounce amber glass prescription bottles in the dark at 4 degrees C. Immediately after preparation and at 3, 7, 14, 21, and 28 days, samples were visually inspected, tested for pH, and assayed in duplicate by high-performance liquid chromatography. On day 28, the mean percentages of the initial clonidine hydrochloride concentrations remaining were 92.4% in the suspension and 93.7% in the solution. The color, odor, and pH of the samples did not change appreciably over the study period. An extemporaneously compounded oral liquid preparation of clonidine hydrochloride in Simple Syrup, NF, is stable under the conditions studied for up to 28 days.

UI MeSH Term Description Entries
D002851 Chromatography, High Pressure Liquid Liquid chromatographic techniques which feature high inlet pressures, high sensitivity, and high speed. Chromatography, High Performance Liquid,Chromatography, High Speed Liquid,Chromatography, Liquid, High Pressure,HPLC,High Performance Liquid Chromatography,High-Performance Liquid Chromatography,UPLC,Ultra Performance Liquid Chromatography,Chromatography, High-Performance Liquid,High-Performance Liquid Chromatographies,Liquid Chromatography, High-Performance
D003000 Clonidine An imidazoline sympatholytic agent that stimulates ALPHA-2 ADRENERGIC RECEPTORS and central IMIDAZOLINE RECEPTORS. It is commonly used in the management of HYPERTENSION. Catapres,Catapresan,Catapressan,Chlophazolin,Clofelin,Clofenil,Clonidine Dihydrochloride,Clonidine Hydrochloride,Clonidine Monohydrobromide,Clonidine Monohydrochloride,Clopheline,Dixarit,Gemiton,Hemiton,Isoglaucon,Klofelin,Klofenil,M-5041T,ST-155,Dihydrochloride, Clonidine,Hydrochloride, Clonidine,M 5041T,M5041T,Monohydrobromide, Clonidine,Monohydrochloride, Clonidine,ST 155,ST155
D004339 Drug Compounding The preparation, mixing, and assembly of a drug. (From Remington, The Science and Practice of Pharmacy, 19th ed, p1814). Drug Formulation,Drug Preparation,Drug Microencapsulation,Pharmaceutical Formulation,Compounding, Drug,Formulation, Drug,Formulation, Pharmaceutical,Microencapsulation, Drug,Preparation, Drug
D004355 Drug Stability The chemical and physical integrity of a pharmaceutical product. Drug Shelf Life,Drugs Shelf Lives,Shelf Life, Drugs,Drug Stabilities,Drugs Shelf Life,Drugs Shelf Live,Life, Drugs Shelf,Shelf Life, Drug,Shelf Live, Drugs,Shelf Lives, Drugs
D013535 Suspensions Colloids with liquid continuous phase and solid dispersed phase; the term is used loosely also for solid-in-gas (AEROSOLS) and other colloidal systems; water-insoluble drugs may be given as suspensions. Suspension

Related Publications

M L Levinson, and C E Johnson
July 1992, American journal of hospital pharmacy,
M L Levinson, and C E Johnson
November 1993, American journal of hospital pharmacy,
M L Levinson, and C E Johnson
January 1995, American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists,
M L Levinson, and C E Johnson
May 2002, American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists,
M L Levinson, and C E Johnson
February 1991, American journal of hospital pharmacy,
M L Levinson, and C E Johnson
May 1996, American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists,
M L Levinson, and C E Johnson
February 1994, American journal of hospital pharmacy,
M L Levinson, and C E Johnson
October 1994, American journal of hospital pharmacy,
M L Levinson, and C E Johnson
November 1999, American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists,
M L Levinson, and C E Johnson
July 2000, American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists,
Copied contents to your clipboard!