Oxidation of 5,8,11,14,17-eicosapentaenoic acid by hepatic and renal microsomes. 1988

M Van Rollins, and P D Frade, and O A Carretero
Hypertension Research, Division Henry Ford Hospital, Detroit, MI 48202.

Liver and kidney microsomes were isolated from rats raised on high-fat diets. In terms of energy, the high-fat diets contained 4% vegetable and 40% fish, vegetable or coconut oils. Each microsomal preparation was fortified with 1 mM NADPH and incubated with 5,8,11,14,17-eicosapentaenoic acid (20:5(n-3]. The number of metabolites formed was assessed by reverse-phase high-performance liquid chromatography (HPLC). To identify the major metabolites, large-scale incubations were done with 20:5(n-3) and microsomes from phenobarbital-treated rats. After extracts from the phenobarbital and dietary studies were combined, individual products were isolated by reverse- and normal-phase HPLC. The metabolites were identified by mass spectrometry, by chromatographic properties, and by comparing their retention times and mass spectra with those of chemically synthesized standards. For liver microsomes, the major metabolites were: 17,18-, 14,15-, 11,12- and 8,9-dihydroxyeicosatetraenoic acids, 20-hydroxyeicosapentaenoic acid, and 19-hydroxyeicosatetraenoic acid. For renal microsomes, the major metabolites were 20-hydroxyeicosapentaenoic and 19-hydroxypentaenoic acids. Because formation of these metabolites required NADPH and was enhanced by phenobarbital pretreatment, 20:5(n-3) appears to be oxidized by cytochrome P-450 monooxygenases. Based on reverse-phase high performance liquid chromatograms, all three high-fat diets may produce the same types of monooxygenase metabolites from 20:5(n-3). It remains unknown whether fish-oil diets induce the synthesis of monooxygenases to oxidize n-3 fatty acids, because these preliminary studies involved only two animals per dietary group.

UI MeSH Term Description Entries
D007668 Kidney Body organ that filters blood for the secretion of URINE and that regulates ion concentrations. Kidneys
D008099 Liver A large lobed glandular organ in the abdomen of vertebrates that is responsible for detoxification, metabolism, synthesis and storage of various substances. Livers
D008861 Microsomes Artifactual vesicles formed from the endoplasmic reticulum when cells are disrupted. They are isolated by differential centrifugation and are composed of three structural features: rough vesicles, smooth vesicles, and ribosomes. Numerous enzyme activities are associated with the microsomal fraction. (Glick, Glossary of Biochemistry and Molecular Biology, 1990; from Rieger et al., Glossary of Genetics: Classical and Molecular, 5th ed) Microsome
D008862 Microsomes, Liver Closed vesicles of fragmented endoplasmic reticulum created when liver cells or tissue are disrupted by homogenization. They may be smooth or rough. Liver Microsomes,Liver Microsome,Microsome, Liver
D010084 Oxidation-Reduction A chemical reaction in which an electron is transferred from one molecule to another. The electron-donating molecule is the reducing agent or reductant; the electron-accepting molecule is the oxidizing agent or oxidant. Reducing and oxidizing agents function as conjugate reductant-oxidant pairs or redox pairs (Lehninger, Principles of Biochemistry, 1982, p471). Redox,Oxidation Reduction
D010634 Phenobarbital A barbituric acid derivative that acts as a nonselective central nervous system depressant. It potentiates GAMMA-AMINOBUTYRIC ACID action on GABA-A RECEPTORS, and modulates chloride currents through receptor channels. It also inhibits glutamate induced depolarizations. Phenemal,Phenobarbitone,Phenylbarbital,Gardenal,Hysteps,Luminal,Phenobarbital Sodium,Phenobarbital, Monosodium Salt,Phenylethylbarbituric Acid,Acid, Phenylethylbarbituric,Monosodium Salt Phenobarbital,Sodium, Phenobarbital
D004042 Dietary Fats, Unsaturated Unsaturated fats or oils used in foods or as a food. Dietary Oils,Unsaturated Dietary Fats,Dietary Fat, Unsaturated,Dietary Oil,Fat, Unsaturated Dietary,Fats, Unsaturated Dietary,Oil, Dietary,Oils, Dietary,Unsaturated Dietary Fat
D004790 Enzyme Induction An increase in the rate of synthesis of an enzyme due to the presence of an inducer which acts to derepress the gene responsible for enzyme synthesis. Induction, Enzyme
D005395 Fish Oils Oils high in unsaturated fats extracted from the bodies of fish or fish parts, especially the LIVER. Those from the liver are usually high in VITAMIN A. The oils are used as DIETARY SUPPLEMENTS. They are also used in soaps and detergents and as protective coatings. Fish Liver Oils,Fish Oil,Liver Oils, Fish,Oil, Fish,Oils, Fish,Oils, Fish Liver
D000818 Animals Unicellular or multicellular, heterotrophic organisms, that have sensation and the power of voluntary movement. Under the older five kingdom paradigm, Animalia was one of the kingdoms. Under the modern three domain model, Animalia represents one of the many groups in the domain EUKARYOTA. Animal,Metazoa,Animalia

Related Publications

M Van Rollins, and P D Frade, and O A Carretero
January 1981, Progress in lipid research,
M Van Rollins, and P D Frade, and O A Carretero
June 1980, Biochimica et biophysica acta,
M Van Rollins, and P D Frade, and O A Carretero
February 1987, British journal of pharmacology,
M Van Rollins, and P D Frade, and O A Carretero
September 1979, Prostaglandins,
M Van Rollins, and P D Frade, and O A Carretero
July 1989, Nihon yakurigaku zasshi. Folia pharmacologica Japonica,
M Van Rollins, and P D Frade, and O A Carretero
June 1968, Science (New York, N.Y.),
M Van Rollins, and P D Frade, and O A Carretero
January 1981, Progress in lipid research,
M Van Rollins, and P D Frade, and O A Carretero
June 1987, Naunyn-Schmiedeberg's archives of pharmacology,
M Van Rollins, and P D Frade, and O A Carretero
October 1974, Biochemical and biophysical research communications,
M Van Rollins, and P D Frade, and O A Carretero
January 1998, Medical hypotheses,
Copied contents to your clipboard!