Influence of zopiclone on male reproductivity in rats. 1987

T Umemura, and K Yamaguchi, and M Watanabe, and K Esaki, and H Kawamoto, and T Yanagita

The influence of zopiclone, a non-benzodiazepine hypnotic, on male reproductivity and the recovery of the influences were examined in rats since it was found that oral administration of zopiclone to male rats produced sperm death and infertility at doses of 50 mg/kg or more. In the present study, zopiclone was administered orally by gavage at doses of 50 and 250 mg/kg once daily for 6 weeks to male rats of 8 weeks old. The rats were paired with untreated female rats at the end of the 2nd, 4th, and 6th weeks of administration and of the 2nd, 4th, and 6th weeks after termination of the administration. As the results, the copulation rates were 100% in the 50 mg/kg group, but the rate was low in the 250 mg/kg group at the end of the 2nd week of administration. The pregnancy rates of 0% and low motility and morphological abnormalities of the sperm were observed in the zopiclone-treated groups at the end of the 2nd week of administration. In the histological examination of the male reproductive organs, such changes as arrest of spermatogenesis and dilation of the epididymal ducts filled with the sperm were observed in the 250 mg/kg group at the end of the 2nd week of administration. In the recovery observation, the ability to impregnate female rats and the condition of the sperm recovered in the 50 mg/kg group at the end of the 2nd week of recovery. In the most rats of the 250 mg/kg group the ability to impregnate female rats and the condition of the sperm recovered at the end of the 4th and 6th weeks of recovery. However, in some rats of the 250 mg/kg group the ability to impregnate female rats and the condition of the sperm were still not recovered at the end of the 6th week of recovery.

UI MeSH Term Description Entries
D006993 Hypnotics and Sedatives Drugs used to induce drowsiness or sleep or to reduce psychological excitement or anxiety. Hypnotic,Sedative,Sedative and Hypnotic,Sedatives,Hypnotic Effect,Hypnotic Effects,Hypnotics,Sedative Effect,Sedative Effects,Sedatives and Hypnotics,Effect, Hypnotic,Effect, Sedative,Effects, Hypnotic,Effects, Sedative,Hypnotic and Sedative
D008297 Male Males
D010879 Piperazines Compounds that are derived from PIPERAZINE.
D011247 Pregnancy The status during which female mammals carry their developing young (EMBRYOS or FETUSES) in utero before birth, beginning from FERTILIZATION to BIRTH. Gestation,Pregnancies
D011919 Rats, Inbred Strains Genetically identical individuals developed from brother and sister matings which have been carried out for twenty or more generations or by parent x offspring matings carried out with certain restrictions. This also includes animals with a long history of closed colony breeding. August Rats,Inbred Rat Strains,Inbred Strain of Rat,Inbred Strain of Rats,Inbred Strains of Rats,Rat, Inbred Strain,August Rat,Inbred Rat Strain,Inbred Strain Rat,Inbred Strain Rats,Inbred Strains Rat,Inbred Strains Rats,Rat Inbred Strain,Rat Inbred Strains,Rat Strain, Inbred,Rat Strains, Inbred,Rat, August,Rat, Inbred Strains,Rats Inbred Strain,Rats Inbred Strains,Rats, August,Rats, Inbred Strain,Strain Rat, Inbred,Strain Rats, Inbred,Strain, Inbred Rat,Strains, Inbred Rat
D012098 Reproduction The total process by which organisms produce offspring. (Stedman, 25th ed) Human Reproductive Index,Human Reproductive Indexes,Reproductive Period,Human Reproductive Indices,Index, Human Reproductive,Indexes, Human Reproductive,Indices, Human Reproductive,Period, Reproductive,Periods, Reproductive,Reproductive Index, Human,Reproductive Indices, Human,Reproductive Periods
D001835 Body Weight The mass or quantity of heaviness of an individual. It is expressed by units of pounds or kilograms. Body Weights,Weight, Body,Weights, Body
D005260 Female Females
D005837 Genitalia, Male The male reproductive organs. They are divided into the external organs (PENIS; SCROTUM; and URETHRA) and the internal organs (TESTIS; EPIDIDYMIS; VAS DEFERENS; SEMINAL VESICLES; EJACULATORY DUCTS; PROSTATE; and BULBOURETHRAL GLANDS). Accessory Sex Organs, Male,Genital Organs, Male,Sex Organs, Accessory, Male,Genitals, Male,Reproductive System, Male,Genital, Male,Male Genital,Male Genital Organs,Male Genitalia,Male Genitals,Male Reproductive System,Male Reproductive Systems,Reproductive Systems, Male
D000818 Animals Unicellular or multicellular, heterotrophic organisms, that have sensation and the power of voluntary movement. Under the older five kingdom paradigm, Animalia was one of the kingdoms. Under the modern three domain model, Animalia represents one of the many groups in the domain EUKARYOTA. Animal,Metazoa,Animalia

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