Effect of antacids on salicylate kinetics. 1985

R A Shastri

The effect of an antacid on the absorption of aspirin can vary depending on certain physical characteristics of the brand of aspirin chosen. In a study carried out to test the effect of a commonly used antacid on the absorption of a brand of aspirin, no differences were seen in the area under the curve (AUC) of plasma concentrations of salicylic acid versus time, Cmax and Ka of salicylic acid without or with antacid. However, the antacid was seen to alter the pH of urine in four of the six subjects investigated. The study, when extended to examine the effect of antacid on steady-state kinetics of salicylic acid, showed that when the Cmin plasma concentrations of salicylic acid were in the region of 15 mg%, the antacid reduced the plasma concentrations and half-life of salicylic acid. It therefore follows that 15 mg% is the minimum plasma concentration at which an antacid that alters the pH of urine brings about a reduction in the steady-state plasma concentrations and an increase in the elimination of salicylic acid from plasma.

UI MeSH Term Description Entries
D007408 Intestinal Absorption Uptake of substances through the lining of the INTESTINES. Absorption, Intestinal
D007700 Kinetics The rate dynamics in chemical or physical systems.
D008276 Magnesium Hydroxide An inorganic compound that occurs in nature as the mineral brucite. It acts as an antacid with cathartic effects. Brucite,Magnesium Hydrate,Magnesium Hydroxide (Mg(OH)4),Hydrate, Magnesium,Hydroxide, Magnesium
D008297 Male Males
D004338 Drug Combinations Single preparations containing two or more active agents, for the purpose of their concurrent administration as a fixed dose mixture. Drug Combination,Combination, Drug,Combinations, Drug
D006801 Humans Members of the species Homo sapiens. Homo sapiens,Man (Taxonomy),Human,Man, Modern,Modern Man
D006863 Hydrogen-Ion Concentration The normality of a solution with respect to HYDROGEN ions; H+. It is related to acidity measurements in most cases by pH pH,Concentration, Hydrogen-Ion,Concentrations, Hydrogen-Ion,Hydrogen Ion Concentration,Hydrogen-Ion Concentrations
D000328 Adult A person having attained full growth or maturity. Adults are of 19 through 44 years of age. For a person between 19 and 24 years of age, YOUNG ADULT is available. Adults
D000536 Aluminum Hydroxide A compound with many biomedical applications: as a gastric antacid, an antiperspirant, in dentifrices, as an emulsifier, as an adjuvant in bacterins and vaccines, in water purification, etc. Hydrated Alumina,Aldrox,Algeldrate,Alhydrogel,Alugel,Amphojel,Basalgel,Brasivil,Dialume,Nephrox,Pepsamer,Rocgel,Alumina, Hydrated,Hydroxide, Aluminum
D000863 Antacids Substances that counteract or neutralize acidity of the GASTROINTESTINAL TRACT. Alkalinizing Agent,Antacid,Alkalinizing Agents,Agent, Alkalinizing,Agents, Alkalinizing

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