Pharmacokinetics of furosemide urinary elimination by nephrotic children. 1983

J Prandota

Single doses of 2 mg/kg of furosemide (F) were given postprandially as tablets to 17 steroid-responsive nephrotic syndrome (NS) patients, 2.5-15 years old, and seven control children requiring F therapy. One-half, 1, and 2 h after administration, F absorption rate, calculated from the drug urinary excretion data, was significantly more rapid in the NS patients compared to that in the controls. Bioavailability of F in the nephrotic children averaged 58.8% indicating that the gastrointestinal absorption of the drug was unaffected by the disease and by the age of the patients. The first pass effect of F was 24% of the administered dose. The elimination half-life of F, calculated from the drug urinary excretion data in the NS patients was 2.06 +/- 0.96 h (mean +/- SD), whereas in the control children, it was 2.14 +/- 0.69 h. There seems to be no relationship between F elimination half-life and the serum albumin concentration in the NS patients. Also, no correlation was found between the amount of F (mg) excreted in urine during 2 or 6 h after administration (the time of complete absorption of F from the gastrointestinal tract, and the time of the drug diuretic effect, respectively) and the serum albumin concentration in the NS patients. Moreover, no significant difference in the cumulative F urinary excretion was found between both groups of children. The data indicate that factors in addition to serum albumin concentration play a role in the elimination kinetics of F in nephrotic children.

UI MeSH Term Description Entries
D007408 Intestinal Absorption Uptake of substances through the lining of the INTESTINES. Absorption, Intestinal
D007700 Kinetics The rate dynamics in chemical or physical systems.
D008297 Male Males
D009404 Nephrotic Syndrome A condition characterized by severe PROTEINURIA, greater than 3.5 g/day in an average adult. The substantial loss of protein in the urine results in complications such as HYPOPROTEINEMIA; generalized EDEMA; HYPERTENSION; and HYPERLIPIDEMIAS. Diseases associated with nephrotic syndrome generally cause chronic kidney dysfunction. Childhood Idiopathic Nephrotic Syndrome,Frequently Relapsing Nephrotic Syndrome,Multi-Drug Resistant Nephrotic Syndrome,Pediatric Idiopathic Nephrotic Syndrome,Steroid-Dependent Nephrotic Syndrome,Steroid-Resistant Nephrotic Syndrome,Steroid-Sensitive Nephrotic Syndrome,Multi Drug Resistant Nephrotic Syndrome,Nephrotic Syndrome, Steroid-Dependent,Nephrotic Syndrome, Steroid-Resistant,Nephrotic Syndrome, Steroid-Sensitive,Nephrotic Syndromes,Steroid Dependent Nephrotic Syndrome,Steroid Resistant Nephrotic Syndrome,Steroid Sensitive Nephrotic Syndrome,Steroid-Dependent Nephrotic Syndromes,Steroid-Resistant Nephrotic Syndromes,Steroid-Sensitive Nephrotic Syndromes,Syndrome, Nephrotic,Syndrome, Steroid-Sensitive Nephrotic
D002648 Child A person 6 to 12 years of age. An individual 2 to 5 years old is CHILD, PRESCHOOL. Children
D002675 Child, Preschool A child between the ages of 2 and 5. Children, Preschool,Preschool Child,Preschool Children
D005260 Female Females
D005665 Furosemide A benzoic-sulfonamide-furan. It is a diuretic with fast onset and short duration that is used for EDEMA and chronic RENAL INSUFFICIENCY. Frusemide,Fursemide,Errolon,Frusemid,Furanthril,Furantral,Furosemide Monohydrochloride,Furosemide Monosodium Salt,Fusid,Lasix
D006207 Half-Life The time it takes for a substance (drug, radioactive nuclide, or other) to lose half of its pharmacologic, physiologic, or radiologic activity. Halflife,Half Life,Half-Lifes,Halflifes
D006801 Humans Members of the species Homo sapiens. Homo sapiens,Man (Taxonomy),Human,Man, Modern,Modern Man

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