Fate of prostaglandin E2 in suckling rats after intragastric administration. 1982

B Revsin, and R J Lemen, and O Koldovský

[3H]Prostaglandin E2 was administered intragastrically to suckling rats at 10 micrograms and 0.1 microgram doses. At the higher dose, 91% of the radioactive label was recoverable at zero time, decreasing to 29% at 5 h. At the lower dose, 40% of the dose was recoverable at zero time, decreasing to 8% at 5 h. With time, the radioactivity in the stomach showed a steady decrease whereas it increased in the tissues. At the 10 microgram dose of [3H]prostaglandin E2 the amount of radioactivity showed a steady increase in the small intestine lumen and small intestine wall. In liver and kidney the maximum amount of radioactive label was found at 1 h. After 1 h the radioactivity began to decline in the liver, while the kidney remained at the same level for the entire 5-h period. At the 0.1 microgram dose of [3H]prostaglandin E2 the radioactivity in the small intestine lumen reached a maximum 3 h after gavage and thereafter declined. The amount of label in the small intestine wall increased for the entire 5 h. In liver and kidney the radioactivity peaked at 1 h, remained at the same level until the 3rd h, then exhibited a decline. Quantitation of the unmetabolized prostaglandin E2 reaching the various organs studied was possible 30 and 60 min after administration of the 10 micrograms dose of prostaglandin E2. At 30 min 42.9% of radioactive label present in the liver could be shown to be authentic prostaglandin E2. This corresponded to 0.64% of the original dose. At 60 min only 22.8% of the radioactive label found in the liver could be shown to be authentic prostaglandin E2, which corresponded to 0.46% of the administered dose. Similar results were found in the small intestine lumen, the small intestine wall and in the kidney. At 3 and 5h, none of the radioactivity found in these organs could be identified as authentic prostaglandin E2.

UI MeSH Term Description Entries
D007408 Intestinal Absorption Uptake of substances through the lining of the INTESTINES. Absorption, Intestinal
D008297 Male Males
D011458 Prostaglandins E (11 alpha,13E,15S)-11,15-Dihydroxy-9-oxoprost-13-en-1-oic acid (PGE(1)); (5Z,11 alpha,13E,15S)-11,15-dihydroxy-9-oxoprosta-5,13-dien-1-oic acid (PGE(2)); and (5Z,11 alpha,13E,15S,17Z)-11,15-dihydroxy-9-oxoprosta-5,13,17-trien-1-oic acid (PGE(3)). Three of the six naturally occurring prostaglandins. They are considered primary in that no one is derived from another in living organisms. Originally isolated from sheep seminal fluid and vesicles, they are found in many organs and tissues and play a major role in mediating various physiological activities. PGE
D011919 Rats, Inbred Strains Genetically identical individuals developed from brother and sister matings which have been carried out for twenty or more generations or by parent x offspring matings carried out with certain restrictions. This also includes animals with a long history of closed colony breeding. August Rats,Inbred Rat Strains,Inbred Strain of Rat,Inbred Strain of Rats,Inbred Strains of Rats,Rat, Inbred Strain,August Rat,Inbred Rat Strain,Inbred Strain Rat,Inbred Strain Rats,Inbred Strains Rat,Inbred Strains Rats,Rat Inbred Strain,Rat Inbred Strains,Rat Strain, Inbred,Rat Strains, Inbred,Rat, August,Rat, Inbred Strains,Rats Inbred Strain,Rats Inbred Strains,Rats, August,Rats, Inbred Strain,Strain Rat, Inbred,Strain Rats, Inbred,Strain, Inbred Rat,Strains, Inbred Rat
D005260 Female Females
D000818 Animals Unicellular or multicellular, heterotrophic organisms, that have sensation and the power of voluntary movement. Under the older five kingdom paradigm, Animalia was one of the kingdoms. Under the modern three domain model, Animalia represents one of the many groups in the domain EUKARYOTA. Animal,Metazoa,Animalia
D013270 Stomach An organ of digestion situated in the left upper quadrant of the abdomen between the termination of the ESOPHAGUS and the beginning of the DUODENUM. Stomachs
D013997 Time Factors Elements of limited time intervals, contributing to particular results or situations. Time Series,Factor, Time,Time Factor
D014018 Tissue Distribution Accumulation of a drug or chemical substance in various organs (including those not relevant to its pharmacologic or therapeutic action). This distribution depends on the blood flow or perfusion rate of the organ, the ability of the drug to penetrate organ membranes, tissue specificity, protein binding. The distribution is usually expressed as tissue to plasma ratios. Distribution, Tissue,Distributions, Tissue,Tissue Distributions
D014886 Weaning Permanent deprivation of breast milk and commencement of nourishment with other food. (From Stedman, 25th ed) Weanings

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