Adsorptive pinocytosis of phosphorylated oligosaccharides by human fibroblasts. 1982

K E Creek, and W S Sly

Adsorptive pinocytosis of lysosomal enzymes by human fibroblasts depends on phosphomannosyl recognition markers on the enzymes and on high affinity receptors on the cell surface. To define the role of phosphorylated oligosaccharides in enzyme recognition, we studied the pinocytosis of [2-3H]mannose-labeled oligosaccharides purified from glycoproteins secreted by fibroblasts. Uptake of the oligosaccharides was inhibited 97% by 2 mM mannose-6-phosphate, 33% by 2 mM glucose 6-phosphate, and 5% or less by 2 mM alpha-methylmannoside, mannose, galactose, or L-fucose. The oligosaccharides were separated into neutral and five anionic species by chromatography on quaternary aminoethyl-Sephadex, characterized, and compared for susceptibility to pinocytosis. Treatment of the phosphorylated oligosaccharides with alkaline phosphatase before or after mild acid hydrolysis demonstrated that they contained one or two phosphates in phosphodiester linkage (covered) or phosphomonoester linkage (uncovered), or two phosphates, one in monoester linkage and one in diester linkage. Neutral oligosaccharides and those with one covered phosphate were not taken up by fibroblasts. Species with one uncovered phosphate or two covered phosphates showed low but detectable uptake. Oligosaccharides isolated as species with two uncovered phosphates, or those converted to this form by mild acid hydrolysis, were taken up 30-fold greater than the lower uptake forms during a 12-h incubation. Thus, oligosaccharides with two uncovered phosphates were far better ligands for the phosphomannosyl receptor than other oligosaccharides on acid hydrolases secreted by fibroblasts and initial rates of uptake of these oligosaccharides were comparable to those reported for several "high uptake" lysosomal enzymes.

UI MeSH Term Description Entries
D007700 Kinetics The rate dynamics in chemical or physical systems.
D009844 Oligosaccharides Carbohydrates consisting of between two (DISACCHARIDES) and ten MONOSACCHARIDES connected by either an alpha- or beta-glycosidic link. They are found throughout nature in both the free and bound form. Oligosaccharide
D010766 Phosphorylation The introduction of a phosphoryl group into a compound through the formation of an ester bond between the compound and a phosphorus moiety. Phosphorylations
D010873 Pinocytosis The engulfing of liquids by cells by a process of invagination and closure of the cell membrane to form fluid-filled vacuoles. Pinocytoses
D002478 Cells, Cultured Cells propagated in vitro in special media conducive to their growth. Cultured cells are used to study developmental, morphologic, metabolic, physiologic, and genetic processes, among others. Cultured Cells,Cell, Cultured,Cultured Cell
D005347 Fibroblasts Connective tissue cells which secrete an extracellular matrix rich in collagen and other macromolecules. Fibroblast
D006020 Glycopeptides Proteins which contain carbohydrate groups attached covalently to the polypeptide chain. The protein moiety is the predominant group with the carbohydrate making up only a small percentage of the total weight. Glycopeptide
D006600 Hexosephosphates
D006601 Hexoses MONOSACCHARIDES whose molecules contain six carbon atoms, such as GLUCOSE and FRUCTOSE. They generally have the chemical formula C6H12O6. Hexose
D006801 Humans Members of the species Homo sapiens. Homo sapiens,Man (Taxonomy),Human,Man, Modern,Modern Man

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