Facilitation of self-stimulation in rats by methadone. 1980

R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan

The effects of morphine and its derivatives on self-stimulation behavior have been widely studied. In those experiments which have used multiple injections (over days) and multiple post-injection tests (within days), the typical findings includes a depression of responding after the initial injections followed by a facilitation of responding on subsequent days. There have been only a few reports which have tested the effects of methadone in this paradigm. Some investigators have observed only depression of self-stimulation while others have reported both the transient depression and the subsequent facilitation generally obtained with morphine. In the present experiment we administered either 5 mg/kg or 10 mg/kg methadone IP over a five day period and tested MFB-LH self-stimulation at 2, 4, 6, 8, 10 and 23 hours post-injection. Compared to saline controls, the 10 mg/kg dose produced the typical opiate-induced changes in self-stimulation, i.e., an initial depression which lasted for two hours on the first two days but was replaced by significant facilitation by hour 4 of day 3. This facilitation persisted for at least 10 hours on all 5 days of the experiment. Except for a transient (days 2-3) depression of self-stimulation, 5 mg/kg was without effects. The present experiment demonstrates that methadone does facilitate self-stimulation but that its ability to do so is highly dose-dependent.

UI MeSH Term Description Entries
D008297 Male Males
D008691 Methadone A synthetic opioid that is used as the hydrochloride. It is an opioid analgesic that is primarily a mu-opioid agonist. It has actions and uses similar to those of MORPHINE. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1082-3) Amidone,Biodone,Dolophine,Metadol,Metasedin,Methaddict,Methadone Hydrochloride,Methadose,Methex,Phenadone,Phymet,Physeptone,Pinadone,Symoron,Hydrochloride, Methadone
D004361 Drug Tolerance Progressive diminution of the susceptibility of a human or animal to the effects of a drug, resulting from its continued administration. It should be differentiated from DRUG RESISTANCE wherein an organism, disease, or tissue fails to respond to the intended effectiveness of a chemical or drug. It should also be differentiated from MAXIMUM TOLERATED DOSE and NO-OBSERVED-ADVERSE-EFFECT LEVEL. Drug Tolerances,Tolerance, Drug,Tolerances, Drug
D000818 Animals Unicellular or multicellular, heterotrophic organisms, that have sensation and the power of voluntary movement. Under the older five kingdom paradigm, Animalia was one of the kingdoms. Under the modern three domain model, Animalia represents one of the many groups in the domain EUKARYOTA. Animal,Metazoa,Animalia
D012653 Self Stimulation The act or process of inducing or increasing the level of arousal in oneself. It can be observed in various situations; for example, infants who are understimulated may explore their surroundings or babble to themselves.(https://dictionary.apa.org/self-stimulation accessed 12/30/2020) ICSS Intracranial Self-Stimulation,Intracranial Self Stimulation,Self-Stimulation,Intracranial Self Stimulations,Self Stimulation, Intracranial,Self Stimulations,Self Stimulations, Intracranial,Self-Stimulations,Stimulation, Self,Stimulations, Self
D051381 Rats The common name for the genus Rattus. Rattus,Rats, Laboratory,Rats, Norway,Rattus norvegicus,Laboratory Rat,Laboratory Rats,Norway Rat,Norway Rats,Rat,Rat, Laboratory,Rat, Norway,norvegicus, Rattus

Related Publications

R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan
January 1974, Japanese journal of pharmacology,
R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan
November 2010, Hormones and behavior,
R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan
June 1978, Canadian journal of psychology,
R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan
October 2012, Physiology & behavior,
R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan
March 1973, Physiology & behavior,
R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan
January 1969, Science (New York, N.Y.),
R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan
April 2003, Pharmacology, biochemistry, and behavior,
R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan
August 1980, Physiology & behavior,
R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan
May 1984, Physiology & behavior,
R M Stutz, and A N Maroli, and W K Tsang, and P A Harvan
May 1997, Neurobiology of learning and memory,
Copied contents to your clipboard!