5-Formyl- and 10-formyl-5,6,7,8-tetrahydrofolate. Conformation of the tetrahydropyrazine ring and formyl group in solution. 1980

M Poe, and S J Benkovic

The chemical shifts and spin-spin coupling constants for the 300-MHz 1H NMR spectra of (6RS)-10-formyl-and (6RS)-5-formyl-5,6,7,8-tetrahydro-L-folate at 25 degrees C in 0.1 M NaOD and at neutral pH are reported and analyzed. Assignments of most resonances are based on comparison to closely related compounds; the resonances of C(6)-H, C-(7)-2H, and C(9)-2H are assigned by preparation of specifically deuterated formyltetrahydrofolates. From analysis of the C(7)-2H spin-spin coupling constants, it is proposed that the tetrahydropyrazine rings of both 10-formyl- and 5-formyl-H4folate are in a half-chair conformation with C(6)-H equatorial. It is further proposed from model building that the 5-formyl group and C(9) of 5-formyl-H4folate are trans. In the 1H NMR spectrum of 5-CHO-H4folate, there was a minor species which was present at a concentration roughly one-sixth that of the major species; this species did not correspond to oxidized 5-CHO-H4folate and could not be separated from the major species by gel permeation or ion-exchange chromatography. It is proposed that this minor species corresponds to a conformer of 5-CHO-H4folate in slow exchange with the major conformer; this slow exchange is attributed to slow rotation due to a partial double bond character of the N(5) to 5-formyl-carbon bond. During the preparation of 10-formyl-H4folate from 5,10-methenyl-H4folate in D2O, approximately 60% of the formyl hydrogen was exchanged for deuterium. The equilibrium constant for the interconversion of 5,10-methenyl-H4folate and 10-formyl-H4folate, K' = [5,10-methenyl-H4folate]/([D+][10-formyl-H4folate]), was measured to be (1.4 +/- 0.6) X 10(6) M-1 in D2O at 25 degrees C.

UI MeSH Term Description Entries
D008968 Molecular Conformation The characteristic three-dimensional shape of a molecule. Molecular Configuration,3D Molecular Structure,Configuration, Molecular,Molecular Structure, Three Dimensional,Three Dimensional Molecular Structure,3D Molecular Structures,Configurations, Molecular,Conformation, Molecular,Conformations, Molecular,Molecular Configurations,Molecular Conformations,Molecular Structure, 3D,Molecular Structures, 3D,Structure, 3D Molecular,Structures, 3D Molecular
D009682 Magnetic Resonance Spectroscopy Spectroscopic method of measuring the magnetic moment of elementary particles such as atomic nuclei, protons or electrons. It is employed in clinical applications such as NMR Tomography (MAGNETIC RESONANCE IMAGING). In Vivo NMR Spectroscopy,MR Spectroscopy,Magnetic Resonance,NMR Spectroscopy,NMR Spectroscopy, In Vivo,Nuclear Magnetic Resonance,Spectroscopy, Magnetic Resonance,Spectroscopy, NMR,Spectroscopy, Nuclear Magnetic Resonance,Magnetic Resonance Spectroscopies,Magnetic Resonance, Nuclear,NMR Spectroscopies,Resonance Spectroscopy, Magnetic,Resonance, Magnetic,Resonance, Nuclear Magnetic,Spectroscopies, NMR,Spectroscopy, MR
D002850 Chromatography, Gel Chromatography on non-ionic gels without regard to the mechanism of solute discrimination. Chromatography, Exclusion,Chromatography, Gel Permeation,Chromatography, Molecular Sieve,Gel Filtration,Gel Filtration Chromatography,Chromatography, Size Exclusion,Exclusion Chromatography,Gel Chromatography,Gel Permeation Chromatography,Molecular Sieve Chromatography,Chromatography, Gel Filtration,Exclusion Chromatography, Size,Filtration Chromatography, Gel,Filtration, Gel,Sieve Chromatography, Molecular,Size Exclusion Chromatography
D005575 Formyltetrahydrofolates Tetrahydrofolates which are substituted by a formyl group at either the nitrogen atom in the 5 position or the nitrogen atom in the 10 position. N(5)-Formyltetrahydrofolate is leucovorin (citrovorum factor) while N(10)-formyltetrahydrofolate is an active coenzyme which functions as a carrier of the formyl group in a number of enzymatic reactions. Formyltetrahydrofolic Acids,N(10)-Formyltetrahydrofolate
D012995 Solubility The ability of a substance to be dissolved, i.e. to form a solution with another substance. (From McGraw-Hill Dictionary of Scientific and Technical Terms, 6th ed) Solubilities
D013763 Tetrahydrofolates Compounds based on 5,6,7,8-tetrahydrofolate.

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