Finite element analysis of diffusional drug release from complex matrix systems. II. Factors influencing release kinetics. 1998

X Y Wu, and Y Zhou
Faculty of Pharmacy, University of Toronto, Ontario, Canada. xywu@phm.utoronto.ca

This work concentrated on the analysis of several factors influencing the kinetics of diffusional drug release from complex matrix devices, such as convex tablets and rings, into a finite volume. These factors include initial drug concentration distribution, anisotropic matrix, and time- and concentration-dependent diffusion coefficients. The individual and comprehensive effects of these factors on the release kinetics were investigated by the finite element method. Errors introduced by neglecting drug diffusion through the ends of edges of cylindrical devices were estimated by comparison of the 1-D models with the 2-D cylinder model. The influence of side-wall coating on the accuracy of the prediction of release profiles by the 1-D slab model for cylindrical devices was studied using various coating materials of different permeabilities. The analyses carried out in this work could assist the design of the complex matrix systems required for controlled drug release.

UI MeSH Term Description Entries
D007700 Kinetics The rate dynamics in chemical or physical systems.
D002626 Chemistry, Pharmaceutical Chemistry dealing with the composition and preparation of agents having PHARMACOLOGIC ACTIONS or diagnostic use. Medicinal Chemistry,Chemistry, Pharmaceutic,Pharmaceutic Chemistry,Pharmaceutical Chemistry,Chemistry, Medicinal
D003692 Delayed-Action Preparations Dosage forms of a drug that act over a period of time by controlled-release processes or technology. Controlled Release Formulation,Controlled-Release Formulation,Controlled-Release Preparation,Delayed-Action Preparation,Depot Preparation,Depot Preparations,Extended Release Formulation,Extended Release Preparation,Prolonged-Action Preparation,Prolonged-Action Preparations,Sustained Release Formulation,Sustained-Release Preparation,Sustained-Release Preparations,Timed-Release Preparation,Timed-Release Preparations,Controlled-Release Formulations,Controlled-Release Preparations,Extended Release Formulations,Extended Release Preparations,Slow Release Formulation,Sustained Release Formulations,Controlled Release Formulations,Controlled Release Preparation,Controlled Release Preparations,Delayed Action Preparation,Delayed Action Preparations,Formulation, Controlled Release,Formulations, Controlled Release,Prolonged Action Preparation,Release Formulation, Controlled,Release Formulations, Controlled,Sustained Release Preparation,Timed Release Preparation,Timed Release Preparations
D004058 Diffusion The tendency of a gas or solute to pass from a point of higher pressure or concentration to a point of lower pressure or concentration and to distribute itself throughout the available space. Diffusion, especially FACILITATED DIFFUSION, is a major mechanism of BIOLOGICAL TRANSPORT. Diffusions

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