A study of chloramphenicol distribution and residues in dairy cows. 1978

J F Nouws, and G Ziv

Distribution and residues of chloramphenicol were examined in 29 normal and 15 emergency-slaughtered dairy cows after parenteral injection of 3 chloramphenicol base formulations, using microbiological and chemical assay procedures. Five qualitative test methods for antibiotic residues failed to detect the presence of the drug even in samples collected within 18 hours of treatment at a dose level of 37 mg/kg, and in emergency-slaughtered cows known to have been treated with chloramphenicol before slaughter. The limited usefulness of these methods for the detection of chloramphenicol residues is stressed by observations indicating the presence of chemically measurable concentrations of the drugs (or its metabolites) in the muscle, kidney, liver, bile, and urine 65 hours after treatment. Quantitative microbiological assay procedures for chloramphenicol (sensitivity limits 1.0 microgram/ml tissue fluid) conducted on specimens of kidney and liver samples of cows treated with chloramphenicol (doses approximately 10 to 40 mg/kg intramuscularly) 1/2 ; 1; 3 1/2; 12; 18; 46; and 65 hours earlier were all negative. However, chemical assay procedures (sensitivity limits 0.2 to 3 microgram/ml or mu/g tissue) for chloramphenicol and some of its metabolites detected the drug in these samples as well as in the meat. Chloramphenicol is apparently extensively metabolized in adult bovines. The extended persistence of "chloramphenicol" residues in the carcass is due to the relatively slow elimination rate of the metabolized drug and the poor and slow absorption rate from the intramuscular injection site after treatment, with preparations containing chloramphenicol base dissolved in organic solvents. Examples are given of the predicting of of pre-slaughter carcass withdrawal times on the basis of arbitrary drug tolerance or detection levels.

UI MeSH Term Description Entries
D007668 Kidney Body organ that filters blood for the secretion of URINE and that regulates ion concentrations. Kidneys
D008099 Liver A large lobed glandular organ in the abdomen of vertebrates that is responsible for detoxification, metabolism, synthesis and storage of various substances. Livers
D008460 Meat The edible portions of any animal used for food including cattle, swine, goats/sheep, poultry, fish, shellfish, and game. Meats
D008657 Metabolic Clearance Rate Volume of biological fluid completely cleared of drug metabolites as measured in unit time. Elimination occurs as a result of metabolic processes in the kidney, liver, saliva, sweat, intestine, heart, brain, or other site. Total Body Clearance Rate,Clearance Rate, Metabolic,Clearance Rates, Metabolic,Metabolic Clearance Rates,Rate, Metabolic Clearance,Rates, Metabolic Clearance
D009132 Muscles Contractile tissue that produces movement in animals. Muscle Tissue,Muscle,Muscle Tissues,Tissue, Muscle,Tissues, Muscle
D001826 Body Fluids Liquid components of living organisms. Body Fluid,Fluid, Body,Fluids, Body
D002417 Cattle Domesticated bovine animals of the genus Bos, usually kept on a farm or ranch and used for the production of meat or dairy products or for heavy labor. Beef Cow,Bos grunniens,Bos indicus,Bos indicus Cattle,Bos taurus,Cow,Cow, Domestic,Dairy Cow,Holstein Cow,Indicine Cattle,Taurine Cattle,Taurus Cattle,Yak,Zebu,Beef Cows,Bos indicus Cattles,Cattle, Bos indicus,Cattle, Indicine,Cattle, Taurine,Cattle, Taurus,Cattles, Bos indicus,Cattles, Indicine,Cattles, Taurine,Cattles, Taurus,Cow, Beef,Cow, Dairy,Cow, Holstein,Cows,Dairy Cows,Domestic Cow,Domestic Cows,Indicine Cattles,Taurine Cattles,Taurus Cattles,Yaks,Zebus
D002701 Chloramphenicol An antibiotic first isolated from cultures of Streptomyces venequelae in 1947 but now produced synthetically. It has a relatively simple structure and was the first broad-spectrum antibiotic to be discovered. It acts by interfering with bacterial protein synthesis and is mainly bacteriostatic. (From Martindale, The Extra Pharmacopoeia, 29th ed, p106) Cloranfenicol,Kloramfenikol,Levomycetin,Amphenicol,Amphenicols,Chlornitromycin,Chlorocid,Chloromycetin,Detreomycin,Ophthochlor,Syntomycin
D005260 Female Females
D005504 Food Analysis Measurement and evaluation of the components of substances to be taken as FOOD. Analysis, Food,Analyses, Food,Food Analyses

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